2-Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure–Activity Relationships, Mechanism of Action and Absorption, Distribution, Metabolism, and Excretion Characterization | ACS Infectious ...
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8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors | Journal of Medicinal Chemistry
Identification of Imidazo-Pyrrolopyridines as Novel and Potent JAK1 Inhibitors | Journal of Medicinal Chemistry
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Discovery of Potent and Selective Pyrazolopyrimidine Janus Kinase 2 Inhibitors | Journal of Medicinal Chemistry